SCHEMBL28540922

SCHEMBL28540922

COC(=O)c1cc(Br)c(CNC(=O)OC(C)(C)C)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.40
AAK1 Q2M2I8 4/20 0.38
KDM4A O75164 1/20 0.38
ATR Q13535 1/20 0.38
KCNA5 P22460 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
SERPINE1 P05121 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
BDKRB1 P46663 2/20 0.35
EPAS1 Q99814 1/20 0.35
HDAC10 Q969S8 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28542535 0.85 ATR (0.45) SOS1KDM4AATRKCNA5MTNR1A
SCHEMBL28542639 0.81 SCN9A (0.39) KDM4AATRKCNA5CA12CA1
SCHEMBL31706166 0.81 CACNA1H (0.45) AAK1KDM4AKCNA5CA12CA1
SCHEMBL25574990 0.80 AAK1 (0.49) AAK1KDM4AKCNA5MTNR1AMTNR1B
SCHEMBL25215120 0.79 KCNA5 (0.39) AAK1KDM4AATRKCNA5MTNR1A
SCHEMBL24502884 0.78 NOTUM (0.40) SOS1AAK1KDM4AATRKCNA5
SCHEMBL29533276 0.78 AAK1 (0.45) AAK1KDM4AKCNA5CA12CA1
SCHEMBL31515366 0.78 ATR (0.42) SOS1AAK1ATRCA12CA1
SCHEMBL22664847 0.78 AAK1 (0.45) AAK1KDM4AKCNA5CA12CA1
SCHEMBL12231435 0.78 ATR (0.42) KDM4AATRKCNA5CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107200726-B Pyrrolidine-amide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-04-06 CN disclosed