SCHEMBL2854409

SCHEMBL2854409

Clc1cccc(Cl)c1CCNCc1cccnc1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.59
CYP2D6 P10635 2/20 0.59
CHRM2 P08172 1/20 0.58
HTR5A P47898 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
SCN8A Q9UQD0 1/20 0.49
ALDH1A1 P00352 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CXCR4 P61073 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854473 0.83 TAAR1 (0.50) CYP2D6CYP3A4CYP2C19ALDH1A1HTR2A
SCHEMBL16606308 0.82 CYP1A2 (0.74) CYP1A2CYP2D6CHRM2HTR5ASCN8A
SCHEMBL10561741 0.80 CYP1A2 (0.61) CYP1A2CYP2D6CHRM2HTR5AALDH1A1
SCHEMBL29875178 0.80 CYP1A2 (0.83) CYP1A2CYP2D6CHRM2SCN8AALDH1A1
SCHEMBL19031318 0.80 CYP1A2 (0.83) CYP1A2CYP2D6CHRM2SCN8AALDH1A1
SCHEMBL10859183 0.79 CYP1A2 (0.56) CYP1A2CYP2D6CHRM2HTR5ACYP3A4
SCHEMBL7235869 0.79 CYP1A2 (0.69) CYP1A2CYP2D6CHRM2CYP3A4CYP2C9
SCHEMBL10859125 0.78 SCN8A (0.66) CYP1A2CYP2D6CHRM2HTR5ACYP3A4
SCHEMBL24069916 0.78 CYP1A2 (0.68) CYP1A2CYP2D6CHRM2HTR5AALDH1A1
Hydrochloric Acid SCHEMBL30115033 0.78 CYP1A2 (0.67) CYP1A2CYP2D6CHRM2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed