SCHEMBL2854473

SCHEMBL2854473

Clc1cccc(Cl)c1CCNCc1ccncc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.50
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 1/20 0.46
GLA P06280 1/20 0.46
SLC2A4 P14672 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
KMT2A Q03164 1/20 0.43
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 1/20 0.42
ADRB2 P07550 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854483 0.83 CHRM2 (0.55) TAAR1KDM4ESMN1; SMN2CYP3A4CYP2D6
SCHEMBL2854409 0.83 CYP1A2 (0.59) ALDH1A1CYP3A4CYP2D6CYP2C19HTR2A
SCHEMBL17110149 0.80 SCN8A (0.49) KMT2ACYP3A4CYP2D6CYP2C19ADRB2
SCHEMBL4037480 0.76 CA1 (0.51) KDM4EKMT2ACYP2C19ADRB2GAA
SCHEMBL10557535 0.76 CA12 (0.58) TAAR1ALDH1A1KDM4EGLASMN1; SMN2
SCHEMBL29444840 0.75 MEN1 (0.56) TAAR1ALDH1A1KDM4EGLASLC2A4
SCHEMBL28188921 0.75 GAA (0.74) ALDH1A1KDM4EGLASMN1; SMN2KMT2A
SCHEMBL2857026 0.74 CHRM2 (0.57) ALDH1A1KDM4ESMN1; SMN2KMT2ACYP2D6
SCHEMBL1799518 0.74 CHRM2 (0.45) TAAR1KDM4ECYP3A4CYP2D6CYP2C19
SCHEMBL2852240 0.73 MC5R (0.58) CYP3A4CYP2D6CYP2C19HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed