SCHEMBL28544263

SCHEMBL28544263

O=C(O)c1ccc(C(F)(F)F)cc1OCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.60
RXRB P28702 2/20 0.60
RXRG P48443 2/20 0.60
KDM4E B2RXH2 1/20 0.57
USP2 O75604 1/20 0.57
ALDH1A1 P00352 1/20 0.57
HPGD P15428 1/20 0.57
CYP2C19 P33261 1/20 0.57
HSD17B10 Q99714 1/20 0.57
MRGPRX4 Q96LA9 7/20 0.56
NR4A2 P43354 1/20 0.54
LRRK2 Q5S007 3/20 0.54
HTR2C P28335 1/20 0.53
SLC6A4 P31645 1/20 0.53
HTR2B P41595 1/20 0.53
MCL1 Q07820 1/20 0.53
PTGER1 P34995 1/20 0.53
FOLH1 Q04609 1/20 0.51
PTPN2 P17706 1/20 0.51
PTPN1 P18031 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23226557 0.89 PTPN1 (0.61) RXRARXRBRXRGMRGPRX4MCL1
SCHEMBL19667112 0.89 MCL1 (0.54) RXRARXRBRXRGKDM4EUSP2
SCHEMBL31406760 0.89 RXRA (0.58) RXRARXRBRXRGMRGPRX4NR4A2
SCHEMBL4200632 0.89 LRRK2 (0.63) RXRARXRBRXRGKDM4EALDH1A1
SCHEMBL11768921 0.87 LRRK2 (0.61) RXRARXRBRXRGKDM4EALDH1A1
SCHEMBL21436902 0.87 RXRA (0.56) RXRARXRBRXRGMRGPRX4NR4A2
SCHEMBL28558879 0.86 MRGPRX4 (0.57) RXRARXRBRXRGKDM4EALDH1A1
SCHEMBL2451483 0.84 RXRA (0.58) RXRARXRBRXRGALDH1A1MRGPRX4
SCHEMBL27354625 0.84 LRRK2 (0.55) RXRARXRBRXRGMRGPRX4LRRK2
SCHEMBL27354622 0.84 LRRK2 (0.55) RXRARXRBRXRGMRGPRX4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111995567-B Formamide pyridone iron chelator derivative with potential multi-target anti-AD activity and preparation method and application thereof 浙江工业大学 2022-11-25 CN disclosed
CN-111995567-A Formamide pyridone iron chelator derivative with potential multi-target anti-AD activity and preparation method and application thereof 浙江工业大学 2020-11-27 CN disclosed