SCHEMBL28544866

SCHEMBL28544866

CS(=O)(=O)[C@H](O)C(NC(=O)c1ccccc1)(C(=O)O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
CYP2C9 P11712 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
EPHX1 P07099 1/20 0.37
HDAC3 O15379 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
IDO1 P14902 1/20 0.36
ALOX15 P16050 1/20 0.36
HDAC1 Q13547 1/20 0.36
CA9 Q16790 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28699449 0.70 EPHX2 (0.40) POLBCYP2C9CYP3A4CYP2C19NPSR1
SCHEMBL19272562 0.70 MEN1 (0.43) NPSR1LMNASMN1; SMN2HDAC3CA12
SCHEMBL28849403 0.70 CYP1A2 (0.62) CYP2C19SMN1; SMN2HDAC3CA1HDAC1
SCHEMBL28551769 0.70 CYP1A2 (0.41) CYP2C19SMN1; SMN2HDAC3CA1ALOX15
SCHEMBL28536195 0.70 CYP1A2 (0.41) CYP2C19SMN1; SMN2HDAC3CA1ALOX15
SCHEMBL19272539 0.69 KMT2A (0.52) CYP3A4LMNAHDAC1HDAC2HDAC8
SCHEMBL28849391 0.69 CYP1A2 (0.61) CYP2C19SMN1; SMN2HDAC3CA1HDAC1
SCHEMBL28250190 0.68 POLB (0.54) POLBCYP2C9CYP3A4CYP2C19NPSR1
SCHEMBL3039120 0.68 POLB (0.58) POLBCYP2C9CYP3A4CYP2C19NPSR1
SCHEMBL28250046 0.68 POLB (0.49) POLBCYP2C9CYP3A4CYP2C19NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112321467-A Preparation method of (2S,3R) -p-methylsulfonylphenylserine ethyl ester 苏州开元民生科技股份有限公司 2021-02-05 CN disclosed