SCHEMBL28545142

SCHEMBL28545142

CCc1c(Cl)nc2cc(C(=O)O)ccn12

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
AGTR1 P30556 1/20 0.39
AGTR2 P50052 1/20 0.39
POLB P06746 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
SLC22A12 Q96S37 1/20 0.34
TSHR P16473 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21936047 0.85 KDM4E (0.43) NPC1RAB9AKDM4EAKT1AKT2
SCHEMBL17434280 0.81 HDAC1 (0.44) NPC1RAB9AMEN1KMT2AAGTR1
SCHEMBL22152490 0.81 NPC1 (0.38) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL28555999 0.81 NPC1 (0.38) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL21936303 0.73 POLQ (0.41)
SCHEMBL30447727 0.73 POLQ (0.41)
SCHEMBL10175245 0.72 CDH1 (0.48) NPC1RAB9AKDM4EPOLBAKT1
SCHEMBL15900088 0.72 DNMT1 (0.45) NPC1RAB9AKDM4EMEN1KMT2A
SCHEMBL973778 0.71 TDP1 (0.45) NPC1RAB9AKDM4EMEN1KMT2A
SCHEMBL31190916 0.71 NPC1 (0.43) NPC1RAB9AAKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601745-B Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-06-27 CN disclosed
CN-112601745-A Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2021-04-02 CN disclosed