SCHEMBL28548601

SCHEMBL28548601

COc1cccc(O)c1-c1ccno1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
TP53 P04637 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
TSHR P16473 1/20 0.44
EGFR P00533 1/20 0.43
PIM1 P11309 1/20 0.43
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29788605 1.00 MEN1 (0.47) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL29632578 0.77 KDM4E (0.36) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL24936302 0.77 KDM4E (0.36) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL24977286 0.76 EPHX2 (0.41) KMT2AKDM4EALDH1A1LMNAMAPT
SCHEMBL11022631 0.74 TP53 (0.67) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL23084830 0.73 KDM4E (0.45) KDM4EALDH1A1MAPTCA1GAA
SCHEMBL2093729 0.73 CYP1A2 (0.62) TP53KDM4EALDH1A1CYP3A4HPGD
Hydrochloric Acid SCHEMBL7232145 0.70 MEN1 (0.50) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL7235549 0.69 TP53 (0.53) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL17414696 0.68 TP53 (0.57) MEN1KMT2ATP53KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728945-B 3, 5-disubstituted pyrazole compounds as kinase inhibitors and uses thereof 上海瑛派药业有限公司 2024-01-16 CN disclosed
CN-114728945-A 3, 5-disubstituted pyrazole compounds as kinase inhibitors and application thereof 上海瑛派药业有限公司 2022-07-08 CN disclosed
CN-112457306-A 3, 5-disubstituted pyrazole compounds as kinase inhibitors and application thereof 上海瑛派药业有限公司 2021-03-09 CN disclosed