SCHEMBL28548935

SCHEMBL28548935

O=C(O)c1nc2nc(Nc3cccc(S(=O)(=O)CCO)c3)ncc2cc1-c1ccccc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 6/20 0.41
AURKB Q96GD4 6/20 0.41
GSK3B P49841 6/20 0.41
KDR P35968 6/20 0.41
CDK5 Q00535 6/20 0.41
DCLK1 O15075 5/20 0.41
SYK P43405 5/20 0.41
MAP4K4 O95819 5/20 0.41
LCK P06239 5/20 0.41
CDK1 P06493 5/20 0.41
FGFR1 P11362 5/20 0.41
CDK2 P24941 5/20 0.41
MAPK9 P45984 5/20 0.41
GSK3A P49840 5/20 0.41
NTRK2 Q16620 5/20 0.41
TAOK1 Q7L7X3 5/20 0.41
PDPK1 O15530 4/20 0.41
JAK2 O60674 4/20 0.41
ROCK2 O75116 4/20 0.41
NTRK1 P04629 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417446 0.92 AURKA (0.40) AURKAAURKBGSK3BKDRCDK5
SCHEMBL4414503 0.88 RIPK2 (0.49) AURKAAURKBGSK3BKDRCDK5
SCHEMBL4414385 0.88 CYP2C19 (0.41) AURKAAURKBGSK3BKDRCDK5
SCHEMBL4413220 0.87 CDK1 (0.40) AURKAAURKBGSK3BKDRCDK5
SCHEMBL28562488 0.85 RIPK2 (0.47) FGFR1SRCEGFRRIPK2ACVR1
SCHEMBL4417439 0.85 AURKA (0.39) AURKAAURKBGSK3BKDRCDK5
SCHEMBL14600274 0.84 GSK3B (0.48) AURKAGSK3BCDK2GSK3AIGF1R
SCHEMBL4414392 0.84 RIPK2 (0.41) AURKAAURKBGSK3BKDRCDK5
SCHEMBL4414705 0.84 SYK (0.46) AURKAAURKBGSK3BKDRCDK5
SCHEMBL4413379 0.82 PTK2 (0.44) GSK3BKDRMAP4K4CDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112755193-A Method of treating malignancies with anti-tyrosine kinase inhibitors using dianhydrogalactitol or a derivative thereof 德玛医药 2021-05-07 CN disclosed