SCHEMBL28552133

SCHEMBL28552133

CC(C)(C)OC(=O)NC1CCC(n2ncc3c([N+](=O)[O-])cccc32)CC1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 5/20 0.44
JAK2 O60674 2/20 0.44
DRD2 P14416 5/20 0.41
KDM1A O60341 1/20 0.40
MAOB P27338 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
RET P07949 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KDR P35968 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28552131 1.00 JAK1 (0.44) JAK1JAK2DRD2KDM1AMAOB
SCHEMBL25674514 0.90 KMT2A (0.46) JAK1JAK2DRD2KDM1AMAOB
SCHEMBL30464462 0.90 KMT2A (0.46) JAK1JAK2DRD2KDM1AMAOB
SCHEMBL28542915 0.84 JAK1 (0.47) JAK1JAK2DRD2KDM1AMAOB
SCHEMBL28542917 0.84 JAK1 (0.47) JAK1JAK2DRD2KDM1AMAOB
SCHEMBL30491703 0.83 GPR119 (0.52) ALDH1A1
SCHEMBL14909505 0.82 TDP1 (0.44) L3MBTL1KMT2AALDH1A1
SCHEMBL17619666 0.81 JAK1 (0.43) JAK1JAK2DRD2KDM1AMAOB
SCHEMBL25251022 0.79 GPR119 (0.47)
SCHEMBL17619522 0.77 CKS1B (0.48) JAK1JAK2DRD2KDM1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112585119-A Substituted indoles and methods of use thereof EPIZYME股份有限公司 2021-03-30 CN disclosed