SCHEMBL28554255

SCHEMBL28554255

COC(=O)C1(Br)C=CC=C(c2ccccc2)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
SLC6A3 Q01959 3/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
HTT P42858 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP3A4 P08684 3/20 0.32
TSHR P16473 3/20 0.32
MAPT P10636 3/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP2C9 P11712 1/20 0.32
HDAC4 P56524 2/20 0.31
TACR1 P25103 1/20 0.31
TACR3 P29371 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28737053 0.82 MEN1 (0.39) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL29034607 0.81 DDB1 (0.42) KMT2ASLC6A3SLC6A2L3MBTL1ALDH1A1
SCHEMBL19744662 0.81 MEN1 (0.41) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL3454133 0.80 MEN1 (0.37) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL28695093 0.80 MEN1 (0.37) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL28712291 0.76 KMT2A (0.34) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL31198221 0.74 MEN1 (0.32) MEN1KMT2A
SCHEMBL5581649 0.74 SLC6A3 (0.35) MEN1KMT2ASLC6A3SLC6A2SLC6A4
SCHEMBL7041565 0.73 CHRM3 (0.33) MEN1KMT2ACHRM2CHRM4CHRM5
SCHEMBL28852266 0.72 HDAC4 (0.31) NPC1RAB9AHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112689630-A Novel LXR modulators with bicyclic core moieties 菲尼克斯-FXR股份有限公司 2021-04-20 CN disclosed