SCHEMBL28557486

SCHEMBL28557486

COC(=O)c1ccc(-c2ccccc2)c(Cl)c1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 3/20 0.51
SLC6A4 P31645 2/20 0.51
GABRA1 P14867 2/20 0.45
GABRG2 P18507 2/20 0.45
GABRB3 P28472 2/20 0.45
GABRA3 P34903 2/20 0.45
EGFR P00533 1/20 0.44
GABRA5 P31644 1/20 0.43
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
PDK2 Q15119 1/20 0.43
HTT P42858 2/20 0.42
CLCN2 P51788 1/20 0.42
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 3/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6255108 0.86 SLC6A3 (0.55) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL29109366 0.83 SLC6A3 (0.64) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL27605792 0.80 PDCD1 (0.53) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL29109368 0.80 SLC6A3 (0.62) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL31345282 0.80 SLC6A3 (0.62) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL28548807 0.78 SLC6A3 (0.48) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL29416802 0.78 HTT (0.54) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL28543311 0.77 SLC6A3 (0.44) SLC6A3SLC6A4GABRA1GABRG2GABRB3
SCHEMBL19810438 0.77 ABL1 (0.46) SLC6A3SLC6A4PDK2HTTKMT2A
SCHEMBL8779255 0.76 SLC6A3 (0.51) SLC6A3SLC6A4GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112689630-A Novel LXR modulators with bicyclic core moieties 菲尼克斯-FXR股份有限公司 2021-04-20 CN disclosed