SCHEMBL28557679

SCHEMBL28557679

NCCc1ccccc1Br.O=COCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.59
HTR2A P28223 2/20 0.44
IDO1 P14902 3/20 0.41
GPR52 Q9Y2T5 1/20 0.40
CYP2A6 P11509 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
HRH1 P35367 1/20 0.37
AGXT P21549 1/20 0.37
TRPM8 Q7Z2W7 2/20 0.36
LTA4H P09960 1/20 0.36
PLA2G2A P14555 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethylenediamine SCHEMBL28123362 0.81 IDO1 (0.46) TAAR1HTR2AIDO1CYP2A6SMN1; SMN2
SCHEMBL28924 0.77 IDO1 (0.55) TAAR1IDO1GPR52SMN1; SMN2FFAR1
Hydrazine SCHEMBL27604749 0.77 IDO1 (0.50) IDO1SMN1; SMN2AGXTMAPTALDH1A1
SCHEMBL901056 0.77 TSHR (0.52) IDO1AGXTALDH1A1
SCHEMBL265615 0.77 TAAR1 (1.00) TAAR1HTR2AIDO1GPR52CYP2A6
Benzene SCHEMBL25178056 0.77 TSHR (0.52) IDO1AGXTALDH1A1
SCHEMBL503 0.77 TSHR (0.52) IDO1AGXTALDH1A1
SCHEMBL29423333 0.77 TAAR1 (1.00) TAAR1HTR2AIDO1GPR52CYP2A6
Monoethanolamine SCHEMBL27702227 0.76 IDO1 (0.42) TAAR1HTR2AIDO1CYP2A6SMN1; SMN2
SCHEMBL27606449 0.75 MAOA (0.40) TAAR1HTR2AIDO1CYP2A6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112724084-B Preparation method of (S) -5-bromo-1, 2,3, 4-tetrahydro-N-Boc-isoquinoline-1-carboxylic acid 上海彩迩文生化科技有限公司 2022-04-22 CN claimed
CN-112724084-A Preparation method of (S) -5-bromo-1, 2,3, 4-tetrahydro-N-Boc-isoquinoline-1-carboxylic acid 南京艾普特生物医药有限公司 2021-04-30 CN claimed
CN-112724084-B Preparation method of (S) -5-bromo-1, 2,3, 4-tetrahydro-N-Boc-isoquinoline-1-carboxylic acid 上海彩迩文生化科技有限公司 2022-04-22 CN disclosed
CN-112724084-A Preparation method of (S) -5-bromo-1, 2,3, 4-tetrahydro-N-Boc-isoquinoline-1-carboxylic acid 南京艾普特生物医药有限公司 2021-04-30 CN disclosed