SCHEMBL28558708

SCHEMBL28558708

N=C(Cl)c1ccc(C(F)(F)F)nc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.48
HDAC4 P56524 1/20 0.36
DGAT1 O75907 1/20 0.35
PDE10A Q9Y233 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
GRM4 Q14833 1/20 0.34
CASP3 P42574 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
MLYCD O95822 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28549563 0.98 TRPV4 (0.47) TRPV4HDAC4DGAT1PDE10AMRGPRX4
SCHEMBL5484094 0.81 TRPV4 (0.48) TRPV4KCNH2
SCHEMBL627545 0.81 TRPV4 (0.48) TRPV4HDAC4MRGPRX4TRPV1GRM4
SCHEMBL30395883 0.81 TRPV4 (0.48) TRPV4HDAC4MRGPRX4TRPV1GRM4
Hydrochloric Acid SCHEMBL30936029 0.79 TRPV4 (0.47) TRPV4
Hydrochloric Acid SCHEMBL5125109 0.79 TRPV4 (0.47) TRPV4HDAC4MRGPRX4TRPV1GRM4
Hydrochloric Acid SCHEMBL4394798 0.79 TRPV4 (0.47) TRPV4
Hydrochloric Acid SCHEMBL25304395 0.78 TRPV4 (0.46) TRPV4KCNH2
SCHEMBL2538969 0.78 TRPV4 (0.46) TRPV4HDAC4TRPV1SLC6A3KCNH2
SCHEMBL4248074 0.78 TRPV4 (0.46) TRPV4MRGPRX4TRPV1GRM4CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112739689-B Fluorine-containing pyrimidine compound and method for producing same 优迈特株式会社 2022-06-03 CN disclosed
CN-112739689-A Fluorine-containing pyrimidine compound and method for producing same 优迈特株式会社 2021-04-30 CN disclosed