SCHEMBL28559331

SCHEMBL28559331

CN1CC(=O)Nc2ncnc(-c3ccc(C(=O)N[C@@H](Cc4cccc(F)c4)CN4C(=O)c5ccccc5C4=O)cc3)c21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 4/20 0.37
PIN1 Q13526 3/20 0.35
CACNA1G O43497 2/20 0.34
AKT1 P31749 5/20 0.33
AKT2 P31751 5/20 0.33
AKT3 Q9Y243 5/20 0.33
ROCK2 O75116 2/20 0.33
PRKCA P17252 2/20 0.33
CIT O14578 1/20 0.33
PRKCB P05771 1/20 0.33
PRKACA P17612 1/20 0.33
PRKACB P22694 1/20 0.33
PKN1 Q16512 1/20 0.33
PRKD2 Q9BZL6 1/20 0.33
LMNA P02545 1/20 0.32
GRM5 P41594 2/20 0.32
EGFR P00533 1/20 0.32
PIM1 P11309 1/20 0.32
SYK P43405 1/20 0.32
MAPKAPK2 P49137 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28559335 1.00 ROCK1 (0.37) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28545536 0.94 PIN1 (0.35) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28545535 0.94 PIN1 (0.35) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28559733 0.93 PIN1 (0.33) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28559734 0.93 PIN1 (0.33) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28566460 0.92 AKT1 (0.34) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28545482 0.92 PIN1 (0.32) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28566458 0.92 AKT1 (0.34) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28545485 0.92 PIN1 (0.32) ROCK1PIN1CACNA1GAKT1AKT2
SCHEMBL28554895 0.91 MAPK1 (0.32) ROCK1PIN1AKT1AKT2AKT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112480116-A PKB inhibitors 南京正大天晴制药有限公司 2021-03-12 CN disclosed