SCHEMBL28564336

SCHEMBL28564336

CCOC(=O)c1coc2ccc(Oc3ccncc3C(=O)OCc3ccccc3)cc12

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 15/20 0.62
NMT1 P30419 2/20 0.45
MAOB P27338 1/20 0.43
NMT2 O60551 1/20 0.42
PTGS2 P35354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30254805 1.00 GPBAR1 (0.62) GPBAR1NMT1MAOBNMT2PTGS2
SCHEMBL28561390 0.85 GPBAR1 (0.48) GPBAR1NMT1MAOBNMT2PTGS2
SCHEMBL24470811 0.80 MAOB (0.60) NMT1MAOBNMT2
SCHEMBL30569409 0.80 MAOB (0.60) NMT1MAOBNMT2
SCHEMBL28561020 0.80 GPBAR1 (0.82) GPBAR1
SCHEMBL28555064 0.78 GPBAR1 (0.79) GPBAR1
SCHEMBL28572228 0.78 GPBAR1 (0.74) GPBAR1
SCHEMBL28566927 0.77 GPBAR1 (0.78) GPBAR1
SCHEMBL30254934 0.77 GPBAR1 (1.00) GPBAR1
SCHEMBL28572107 0.77 GPBAR1 (1.00) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112794844-B Ester compound, preparation method and application thereof, and ester soft medicine 中国科学院上海药物研究所 2023-03-21 CN disclosed
CN-112794844-A Ester compound, preparation method and application thereof, and ester soft medicine 中国科学院上海药物研究所 2021-05-14 CN disclosed