SCHEMBL28564451

SCHEMBL28564451

C[C@H](NCCCc1ccc(OCc2ccccc2F)cc1)C(N)=O

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.76
SCN3A Q9NY46 3/20 0.55
MAOB P27338 8/20 0.54
PARP15 Q460N3 1/20 0.53
PARP14 Q460N5 1/20 0.53
PARP10 Q53GL7 1/20 0.53
MAOA P21397 1/20 0.51
SIGMAR1 Q99720 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28564453 1.00 SCN9A (0.76) SCN9ASCN3AMAOBPARP15PARP14
SCHEMBL964122 0.93 SCN9A (0.79) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL962699 0.86 SCN9A (1.00) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL29379049 0.86 SCN9A (1.00) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL67329 0.86 SCN9A (1.00) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL67328 0.86 SCN9A (1.00) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL1697252 0.85 SCN9A (0.98) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL1697253 0.85 SCN9A (0.98) SCN9ASCN3AMAOBPARP15PARP14
SCHEMBL963787 0.83 SCN9A (0.85) SCN9ASCN3AMAOBPARP15PARP14
Ralfinamide SCHEMBL1697229 0.83 SCN9A (0.91) SCN9ASCN3AMAOBPARP15PARP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112716927-B Alpha-amino amide compound and preparation method and application thereof 复旦大学 2022-10-14 CN disclosed
CN-112716927-A Alpha-amino amide compound and preparation method and application thereof 复旦大学 2021-04-30 CN disclosed