SCHEMBL2856691

SCHEMBL2856691

CC(C)Oc1cc2c(C(=O)O)c(-c3ccc(F)cc3)oc2cc1N1CCOCC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 7/20 0.42
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 3/20 0.41
HPGD P15428 2/20 0.41
MAPT P10636 2/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
POLB P06746 1/20 0.38
PRKDC P78527 1/20 0.38
RAF1 P04049 1/20 0.37
BRAF P15056 1/20 0.37
GAA P10253 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ATR Q13535 1/20 0.36
NPC1 O15118 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3544726 0.92 ANO1 (0.43) ANO1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL2845058 0.90 CYP3A4 (0.46) MAPTRAF1BRAFRAB9ASMN1; SMN2
SCHEMBL3541879 0.85 ANO1 (0.40) ANO1ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL2840385 0.83 CYP3A4 (0.46)
SCHEMBL2839923 0.82 CYP3A4 (0.44)
SCHEMBL2840249 0.82 CYP3A4 (0.47)
SCHEMBL2840619 0.82 CYP3A4 (0.47)
SCHEMBL2879661 0.82 CYP3A4 (0.49)
SCHEMBL5496262 0.82 CYP3A4 (0.41)
SCHEMBL5256378 0.82 ANO1 (0.66) ANO1ALDH1A1KDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4537315-B2 2010-09-01 JP claimed
EP-1581207-A4 BENZOFURAN COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATMENT AND PROPHYLAXIS OF HEPATITIS C VIRAL INFECTIONS AND ASSOCIATED DISEASES VIROPHARMA INC (US) 2007-07-25 EP claimed
JP-2006510736-A 2006-03-30 JP claimed
EP-1581207-A2 BENZOFURAN COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATMENT AND PROPHYLAXIS OF HEPATITIS C VIRAL INFECTIONS AND ASSOCIATED DISEASES Viropharma Incorporated (US) 2005-10-05 EP claimed
WO-2004041201-A2 BENZOFURAN COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATMENT AND PROPHYLAXIS OF HEPATITIS C VIRAL INFECTIONS AND ASSOCIATED DISEASES VIROPHARMA INCORPORATED (US) 2004-05-21 WO claimed