SCHEMBL28567741

SCHEMBL28567741

COC(=O)C(Cc1ccc(-c2c(C(F)(F)F)cc(C)n(C)c2=O)c2cccnc12)NC(=O)c1c(F)cc(N2CCOCC2C(F)(F)F)cc1F

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 6/20 0.36
ITGA4 P13612 6/20 0.36
ITGB7 P26010 6/20 0.36
CNR2 P34972 5/20 0.35
PIK3C3 Q8NEB9 2/20 0.33
CNR1 P21554 1/20 0.32
WDR5 P61964 2/20 0.31
HSP90AA1 P07900 1/20 0.30
CXCR3 P49682 1/20 0.30
DGAT2 Q96PD7 1/20 0.30
ATR Q13535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29671090 1.00 ITGB1 (0.36) ITGB1ITGA4ITGB7CNR2PIK3C3
SCHEMBL22031450 1.00 ITGB1 (0.36) ITGB1ITGA4ITGB7CNR2PIK3C3
SCHEMBL21978659 0.94 ITGA4 (0.42) ITGB1ITGA4ITGB7PIK3C3WDR5
SCHEMBL21978664 0.94 ITGA4 (0.42) ITGB1ITGA4ITGB7PIK3C3WDR5
SCHEMBL21978667 0.94 ITGA4 (0.42) ITGB1ITGA4ITGB7PIK3C3WDR5
SCHEMBL22031424 0.92 ITGA4 (0.40) ITGB1ITGA4ITGB7CNR2PIK3C3
SCHEMBL29671123 0.92 ITGA4 (0.40) ITGB1ITGA4ITGB7CNR2PIK3C3
SCHEMBL21957457 0.90 ITGB1 (0.43) ITGB1ITGA4ITGB7PIK3C3
SCHEMBL21957462 0.90 ITGB1 (0.43) ITGB1ITGA4ITGB7PIK3C3
SCHEMBL21957463 0.90 ITGB1 (0.43) ITGB1ITGA4ITGB7PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112969504-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-04-09 CN disclosed
CN-112969504-A Compounds for inhibiting alpha 4 beta 7 integrins 吉利德科学公司 2021-06-15 CN disclosed