SCHEMBL28568152

SCHEMBL28568152

Cc1ccc(N)c(CC(=O)Nc2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
EPHX2 P34913 1/20 0.50
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NLRP3 Q96P20 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HPGD P15428 2/20 0.46
TP53 P04637 1/20 0.46
POLB P06746 1/20 0.45
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3815239 0.84 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19EPHX2
SCHEMBL11641261 0.82 RNF4 (0.54) CYP1A2CYP2D6CYP2C9CYP2C19EPHX2
SCHEMBL5162602 0.81 POLB (0.51) RAB9AEPHX2MEN1KMT2AHDAC3
SCHEMBL22169186 0.81 CYP1A2 (0.65) CYP1A2CYP2D6CYP2C9CYP2C19EPHX2
SCHEMBL5165552 0.81 NLRP3 (0.54) NPC1RAB9ACYP1A2CYP2C19MEN1
SCHEMBL24124271 0.79 MAPT (0.62) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL30522640 0.79 MAPT (0.62) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL11644890 0.79 CYP1A2 (0.48) NPC1RAB9ACYP1A2CYP2D6CYP2C9
SCHEMBL11644204 0.78 PRMT1 (0.58) CYP1A2CYP2D6CYP2C9CYP2C19EPHX2
SCHEMBL27988317 0.77 SRC (0.54) NPC1MEN1KMT2ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778203-B Process for the preparation of 1H-indazole-3-carboxylic acid derivatives and granisetron and lonidamine 兰州交通大学 2022-02-15 CN disclosed
CN-112778203-A Process for the preparation of 1H-indazole-3-carboxylic acid derivatives and granisetron and lonidamine 兰州交通大学 2021-05-11 CN disclosed