SCHEMBL28568415

SCHEMBL28568415

CC(=O)SCCCCCCNC(=O)c1n[nH]c2c1CCc1ccncc1-2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.38
NPC1 O15118 2/20 0.37
NAMPT P43490 6/20 0.37
HDAC3 O15379 4/20 0.36
HDAC4 P56524 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC8 Q9BY41 4/20 0.36
HDAC6 Q9UBN7 4/20 0.36
KDM4E B2RXH2 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
TSHR P16473 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28570148 0.85 NAMPT (0.41) NAAANPC1NAMPTHDAC3HDAC4
SCHEMBL28573673 0.85 HDAC6 (0.46) NAAANPC1NAMPTHDAC3HDAC4
SCHEMBL28575703 0.82 CCNA2 (0.39) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28914562 0.81 HDAC3 (0.36) NAAANPC1NAMPTHDAC3HDAC4
SCHEMBL28574656 0.80 HDAC3 (0.40) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28568974 0.78 HDAC3 (0.35) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28576372 0.78 HDAC3 (0.40) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28582772 0.77 HDAC3 (0.37) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28582693 0.76 HDAC3 (0.33) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28577870 0.73 NPC1 (0.42) NPC1KDM4ETSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN claimed
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN disclosed