SCHEMBL28568465

SCHEMBL28568465

Cc1ccc(C(=O)Nc2cc(C(N)=O)n[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.46
NPC1 O15118 5/20 0.46
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ADORA3 P0DMS8 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
ALDH1A1 P00352 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
TP53 P04637 2/20 0.43
MEN1 O00255 2/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28563324 0.81 SMN1; SMN2 (0.47) RAB9ANPC1ADORA3ADORA2AALDH1A1
SCHEMBL5867451 0.75 CCNA2 (0.49) RAB9ANPC1HDAC1HDAC6ADORA3
SCHEMBL14108088 0.73 JAK2 (0.52) RAB9ANPC1SMN1; SMN2MAPTKMT2A
SCHEMBL5008289 0.73 CCNA2 (0.51) RAB9ANPC1ADORA3ADORA2AADORA1
SCHEMBL14019191 0.71 MAPK1 (0.50) RAB9ANPC1ALDH1A1SMN1; SMN2TP53
SCHEMBL28568338 0.71 MAPT (0.49) ALDH1A1SMN1; SMN2TP53MEN1MAPT
SCHEMBL30683712 0.71 SMN1; SMN2 (0.57) RAB9ANPC1ALDH1A1SMN1; SMN2MEN1
SCHEMBL15359833 0.71 NPC1 (0.51) RAB9ANPC1HDAC1HDAC6MEN1
SCHEMBL13777922 0.70 CCNA2 (0.78) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL5867785 0.70 CCNA2 (0.48) RAB9ANPC1ALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423377-B 5-amino-1H-pyrazole derivative, preparation method and medical application 中国药科大学 2021-06-01 CN disclosed
CN-111423377-A 5-amino-1H-pyrazole derivative, preparation method and medical application 中国药科大学 2020-07-17 CN disclosed