SCHEMBL28569262

SCHEMBL28569262

CC(C)[Si](C(C)C)(C(C)C)n1ccc2cc(-c3ccc(O)cc3)cnc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 3/20 0.44
PDGFRB P09619 2/20 0.42
PDGFRA P16234 2/20 0.42
RIPK1 Q13546 1/20 0.41
USP7 Q93009 2/20 0.38
DYRK1A Q13627 3/20 0.37
DYRK1B Q9Y463 3/20 0.37
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
FTO Q9C0B1 1/20 0.35
MAPK10 P53779 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL522712 0.84 MAP4K4 (0.30) DYRK1ADYRK1B
SCHEMBL28569265 0.80 ESR2 (0.36) ESR2MEN1NPC1RAB9AKMT2A
SCHEMBL417021 0.76 CCR1 (0.40)
SCHEMBL413086 0.75 ENPP3 (0.39)
SCHEMBL4478005 0.75 IRAK4 (0.34)
SCHEMBL29533363 0.72 HTR2C (0.35) NPC1RAB9AABL1EGFRHCK
SCHEMBL12147023 0.72 PARP1 (0.34)
SCHEMBL30643452 0.71 KCNH2 (0.35) MEN1RAB9AKMT2A
SCHEMBL28667672 0.71
SCHEMBL23245974 0.69 ENPP3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112661751-B Heterocyclic compounds as BCL-2 inhibitors 南京天印健华医药科技有限公司 2024-06-14 CN disclosed
CN-112661751-A Heterocyclic compounds as BCL-2 inhibitors 南京天印健华医药科技有限公司 2021-04-16 CN disclosed