SCHEMBL28569440

SCHEMBL28569440

Cc1c(C#N)cccc1-c1cc(C#C[Si](C(C)C)(C(C)C)C(C)C)nc(N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)n1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.34
ADORA2B P29275 3/20 0.33
ADORA1 P30542 1/20 0.33
NISCH Q9Y2I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22304359 0.86 ADORA2A (0.36) ADORA2AADORA2BADORA1NISCH
SCHEMBL22304529 0.82 ADORA2A (0.38) ADORA2AADORA2BADORA1NISCH
SCHEMBL30080281 0.82 ADORA2A (0.38) ADORA2AADORA2BADORA1NISCH
SCHEMBL30080613 0.79 NISCH (0.39) ADORA2AADORA2BADORA1NISCH
SCHEMBL30114630 0.75 ADORA2A (0.46) ADORA2AADORA2BADORA1
SCHEMBL20436371 0.75 ADORA2A (0.46) ADORA2AADORA2BADORA1
SCHEMBL28628129 0.74 ADORA2A (0.39) ADORA2AADORA2BNISCH
SCHEMBL30114734 0.74 ADORA2A (0.39) ADORA2AADORA2BNISCH
SCHEMBL28636992 0.74 NUDT1 (0.34) ADORA2AADORA2BNISCH
SCHEMBL30114810 0.74 NUDT1 (0.34) ADORA2AADORA2BNISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112996783-B 2-aminopyrimidine derivatives, preparation method and application thereof in medicines 江苏恒瑞医药股份有限公司 2022-11-18 CN disclosed
CN-112996783-A 2-aminopyrimidine derivatives, preparation method and application thereof in medicines 江苏恒瑞医药股份有限公司 2021-06-18 CN disclosed