SCHEMBL28573158

SCHEMBL28573158

FC(F)n1ccc2ccncc21

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.45
MAPT P10636 15/20 0.44
CDC7 O00311 1/20 0.42
CDK2 P24941 1/20 0.42
SLC22A12 Q96S37 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31751759 0.85 CDC7 (0.41) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL2230256 0.81 NFATC1 (0.46) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL27647386 0.74 RAPGEF4 (0.37) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL23084376 0.74 SLC6A2 (0.50) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL2127959 0.73 SLC22A12 (0.44) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL13892321 0.71 CDK4 (0.45)
SCHEMBL18821952 0.71 CYP19A1 (0.40) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL1892608 0.69 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2
SCHEMBL18821827 0.69 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2
SCHEMBL255050 0.69 MAPT (0.68) CYP19A1MAPTCDC7CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112279849-A N-difluoromethyl azaindole compound and synthesis method thereof 丽水学院 2021-01-29 CN disclosed