SCHEMBL2858113

SCHEMBL2858113

CCCCCC(=O)N(Cc1ccc([O])cc1)Cc1ccc(C#Cc2ccc(CCCC)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.47
PTPRO Q16827 1/20 0.47
FFAR1 O14842 2/20 0.45
FFAR4 Q5NUL3 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
LTB4R2 Q9NPC1 2/20 0.44
FAAH O00519 1/20 0.41
ALDH1A1 P00352 2/20 0.41
BLM P54132 1/20 0.41
PLK1 P53350 1/20 0.40
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA4 P22748 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854924 0.88 RARB (0.55) PTPN11PTPROFFAR1FFAR4HDAC3
SCHEMBL2855523 0.85 PTPN11 (0.43) PTPN11PTPROFFAR1FFAR4ALDH1A1
SCHEMBL2861907 0.84 PDE6D (0.48) PTPN11PTPROFFAR1FFAR4HDAC3
SCHEMBL1734728 0.83 LTB4R2 (0.53) PTPN11PTPROFFAR1FFAR4LTB4R2
SCHEMBL2853695 0.83 PTPN11 (0.40) PTPN11PTPROFFAR1FFAR4ALDH1A1
SCHEMBL1734774 0.82 PTPN11 (0.66) PTPN11PTPROFFAR1FFAR4LTB4R2
SCHEMBL2853426 0.76 LTB4R2 (0.61) PTPN11PTPROLTB4R2ALDH1A1
SCHEMBL13711743 0.75 RARB (0.71) HDAC3HDAC1HDAC2HDAC6NCOR2
SCHEMBL4398063 0.74 LTB4R2 (0.64) HDAC3HDAC1HDAC2HDAC6NCOR2
SCHEMBL2857121 0.74 S1PR1 (0.45) FFAR1FFAR4ALDH1A1PLK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654247-B1 ALKYNYL ARYL CARBOXAMIDES MERCK SERONO SA (CH) 2010-01-20 EP claimed