SCHEMBL28587194

SCHEMBL28587194

CC(C)(C#N)c1ccnc(Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.42
ROCK2 O75116 3/20 0.42
PRKCQ Q04759 3/20 0.42
PRKCD Q05655 3/20 0.42
ROCK1 Q13464 3/20 0.42
PRKCA P17252 2/20 0.42
PRKACA P17612 1/20 0.42
FLT3 P36888 1/20 0.42
GSK3B P49841 1/20 0.42
JAK3 P52333 1/20 0.42
CSNK1A1 P48729 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
MAPK9 P45984 1/20 0.32
MAPK10 P53779 1/20 0.32
CHRNA7 P36544 1/20 0.32
PIN1 Q13526 1/20 0.31
PDE4A P27815 1/20 0.31
GABRA1 P14867 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31440273 1.00 JAK2 (0.42) JAK2ROCK2PRKCQPRKCDROCK1
SCHEMBL16454353 0.79 JAK2 (0.43) JAK2ROCK2PRKCQPRKCDROCK1
SCHEMBL2018538 0.78 SYK (0.38) GABRA1GABRG2GABRB3GABRA3
SCHEMBL17816271 0.78 JAK2 (0.42) JAK2ROCK2PRKCQPRKCDROCK1
SCHEMBL31543495 0.76 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRA3
SCHEMBL1661164 0.76 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRA3
SCHEMBL30632766 0.75 GABRA1 (0.38) GABRA1GABRG2GABRB3GABRA3
SCHEMBL20015961 0.75 GABRA1 (0.32) GABRA1GABRG2GABRB3GABRA3
SCHEMBL26686630 0.75 GABRA1 (0.38) GABRA1GABRG2GABRB3GABRA3
SCHEMBL2020306 0.75 CYP19A1 (0.37) GABRA1GABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112812105-A Aminopyridyloxypyrazole derivative and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2021-05-18 CN disclosed