SCHEMBL28588229

SCHEMBL28588229

C[C@H](O[C@H]1OCCN[C@H]1c1ccc(F)cc1)c1cc(C(F)F)cc(C(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.39
NR3C1 P04150 1/20 0.39
CYP3A4 P08684 1/20 0.39
FPR1 P21462 1/20 0.39
TACR3 P29371 1/20 0.39
GPR183 P32249 1/20 0.39
OPRD1 P41143 1/20 0.39
GPR65 Q8IYL9 1/20 0.39
GPR35 Q9HC97 1/20 0.39
SCN9A Q15858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28588230 1.00 TACR1 (0.39) TACR1NR3C1CYP3A4FPR1TACR3
Hydrochloric Acid SCHEMBL31593180 0.99 TACR1 (0.39) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL16142417 0.93 TACR1 (0.48) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7022722 0.91 TACR1 (0.41) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7022578 0.89 TACR1 (0.40) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7025187 0.88 TACR1 (0.39) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7025846 0.87 SLC6A2 (0.39) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7023413 0.87 TACR1 (0.39) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7027378 0.86 TACR1 (0.38) TACR1NR3C1CYP3A4FPR1TACR3
SCHEMBL7029570 0.86 ALDH1A1 (0.38) TACR1NR3C1CYP3A4FPR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112939885-A Preparation method of aprepitant key intermediate 海南鑫开源医药科技有限公司 2021-06-11 CN disclosed