SCHEMBL28590003

SCHEMBL28590003

FC(F)(F)c1ccc(O[C@H]2CCCNC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.51
CHRNA4 P43681 2/20 0.51
ROCK1 Q13464 6/20 0.50
ROCK2 O75116 2/20 0.47
PRKX P51817 1/20 0.47
PRKCE Q02156 1/20 0.47
PRKCD Q05655 1/20 0.47
PRKD1 Q15139 1/20 0.47
KCNH2 Q12809 1/20 0.46
HTR2A P28223 1/20 0.46
TIPARP Q7Z3E1 1/20 0.45
SLC6A2 P23975 2/20 0.45
SLC6A4 P31645 1/20 0.45
HTR1A P08908 1/20 0.43
HTR2C P28335 1/20 0.42
CHEK1 O14757 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23166823 1.00 CHRNB2 (0.51) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL28577996 1.00 CHRNB2 (0.51) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL3071569 0.90 SLC6A2 (0.50) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL23791472 0.90 SLC6A2 (0.50) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL23632246 0.90 SLC6A2 (0.50) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL23475081 0.84 CHRNB2 (0.51) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL13761577 0.84 CHRNB2 (0.51) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL3004210 0.83 SLC6A4 (0.49) CHRNB2CHRNA4HTR2ASLC6A2SLC6A4
SCHEMBL19582779 0.82 CHRNB2 (0.55) CHRNB2CHRNA4ROCK1ROCK2PRKX
SCHEMBL15650257 0.82 CHRNB2 (0.55) CHRNB2CHRNA4ROCK1ROCK2PRKX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072521-B ROR gamma t inhibitor and application thereof in medicines 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
CN-113072521-A ROR gamma t inhibitor and application thereof in medicine 广东东阳光药业有限公司 2021-07-06 CN disclosed