SCHEMBL28590804

SCHEMBL28590804

Cn1cc(C(=O)C(=O)Cl)cc1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
POLB P06746 1/20 0.51
TDP1 Q9NUW8 1/20 0.41
PKM P14618 4/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
HDAC8 Q9BY41 1/20 0.34
GPR35 Q9HC97 1/20 0.33
MCL1 Q07820 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GRN P28799 1/20 0.33
SORT1 Q99523 1/20 0.33
USP4 Q13107 1/20 0.32
USP7 Q93009 1/20 0.32
AR P10275 1/20 0.32
GFER P55789 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HDAC10 Q969S8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2783116 0.82 CYP2C9 (0.54) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL17838295 0.81 CYP1A2 (0.55) CYP2C9KMT2AMEN1POLBPKM
SCHEMBL2361283 0.79 CYP2C9 (0.51) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL24158944 0.77 CYP2C9 (0.50) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL27312350 0.76 USP4 (0.51) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL16417130 0.75 CYP2C9 (0.43) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL16416929 0.75 KMT2A (0.43) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL3674837 0.74 TDP1 (0.46) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL1149847 0.73 CYP2C9 (0.60) CYP2C9KMT2AMEN1POLBTDP1
SCHEMBL1277680 0.72 KMT2A (0.53) CYP2C9KMT2AMEN1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108047115-B Glyoxylamide-substituted pyrrole amide derivatives and their use as medicaments for the treatment of hepatitis B 爱尔兰詹森科学公司 2021-06-29 CN disclosed