SCHEMBL28592176

SCHEMBL28592176

C=CCC(NC(=O)OC(C)(C)C)c1cc(-c2ccc(NC(=O)OC)cc2N)ccn1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F11 P03951 3/20 0.38
KLKB1 P03952 2/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
AAK1 Q2M2I8 12/20 0.37
MAP4K4 O95819 1/20 0.35
F10 P00742 1/20 0.34
PLG P00747 1/20 0.34
PLAT P00750 1/20 0.34
HDAC3 O15379 2/20 0.34
SREBF2 Q12772 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL616049 1.00 F11 (0.38) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL616978 0.92 AAK1 (0.34) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL16974676 0.89 F11 (0.42) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL15915827 0.89 F11 (0.38) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL15915824 0.89 F11 (0.38) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL18690161 0.88 AAK1 (0.36) F11AAK1
SCHEMBL18690163 0.88 AAK1 (0.36) F11AAK1
SCHEMBL30193841 0.88 AAK1 (0.36) F11AAK1
SCHEMBL16983835 0.87 AAK1 (0.35) AAK1
SCHEMBL15594121 0.86 AAK1 (0.34) F11AAK1MAP4K4HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108250199-B Dihydropyridone P1 as factor XIA inhibitor 百时美施贵宝公司 2021-07-16 CN disclosed