SCHEMBL28593246

SCHEMBL28593246

[O]CCC1(c2ccccc2)CCc2ccc(Br)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.40
HDAC9 Q9UKV0 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
BACE1 P56817 8/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
APP P05067 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
KDM1B Q8NB78 1/20 0.32
SIGMAR1 Q99720 2/20 0.32
SLC18A3 Q16572 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17748882 0.86 KDM1A (0.40) KDM1AHDAC9OPRM1OPRD1BACE1
SCHEMBL17748895 0.76 BACE1 (0.33) KDM1AOPRM1OPRD1BACE1APP
SCHEMBL11884024 0.64 HDAC9 (0.46) KDM1AHDAC9BACE1MEN1KMT2A
SCHEMBL8708541 0.64 SIGMAR1 (0.41) KDM1AHDAC9MEN1KMT2ASIGMAR1
SCHEMBL27660718 0.64 HDAC9 (0.50) HDAC9BACE1KMT2A
SCHEMBL12077824 0.63 KDM1A (0.55) KDM1ABACE1TDP1L3MBTL1APP
SCHEMBL20449248 0.63 BACE1 (0.48) KDM1ABACE1TDP1L3MBTL1APP
SCHEMBL5709421 0.63 KDM1A (0.43) KDM1AMAOAMAOBSIGMAR1
SCHEMBL9392173 0.63 AKR1B1 (0.51) KDM1ABACE1
SCHEMBL5709333 0.63 KDM1A (0.43) KDM1AMAOAMAOBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107108614-B Substituted pyrrolopyridines as bromodomain inhibitors 基因泰克公司 2021-06-01 CN disclosed