SCHEMBL28598656

SCHEMBL28598656

COc1ccc(N2CCc3ccccc3C2CF)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.48
SLC6A4 P31645 1/20 0.46
DRD2 P14416 3/20 0.46
DRD4 P21917 3/20 0.46
HTR1A P08908 1/20 0.46
HTR1D P28221 1/20 0.46
HTR2A P28223 1/20 0.46
GID4 Q8IVV7 1/20 0.44
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SMPD1 P17405 1/20 0.41
PRMT5 O14744 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28590256 0.84 ESR1 (0.49) HTR2ASIGMAR1MEN1MAPTKMT2A
SCHEMBL12685743 0.81 DRD1 (0.43) DRD1SLC6A4DRD2DRD4HTR1A
SCHEMBL16684242 0.81 DRD1 (0.43) DRD1SLC6A4DRD2DRD4HTR1A
SCHEMBL28451897 0.80 SMPD1 (0.48) DRD1SLC6A4DRD2DRD4HTR1A
SCHEMBL28587854 0.80 HTR3A (0.41) SLC6A4SIGMAR1ALDH1A1HPGD
SCHEMBL28921436 0.76 DRD1 (0.46) DRD1DRD2DRD4HTR1AHTR1D
SCHEMBL29170205 0.75 DRD1 (0.45) DRD1SLC6A4DRD2DRD4HTR1A
SCHEMBL30296945 0.75 DRD1 (0.45) DRD1SLC6A4DRD2DRD4HTR1A
SCHEMBL5525385 0.74 ESR1 (0.62) DRD1DRD2DRD4SIGMAR1DRD5
SCHEMBL28921440 0.74 DRD1 (0.44) DRD1DRD2DRD4HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072493-A Novel synthesis method of 1-fluoromethyl-tetrahydroisoquinoline derivative 中山大学 2021-07-06 CN disclosed