SCHEMBL28598709

SCHEMBL28598709

COC(=O)c1ccc(-c2nc(Nc3cnn(C4CCCNC4)c3)ncc2C)cc1-c1nc(Nc2cnn(C3CCCNC3)c2)ncc1C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.46
AURKB Q96GD4 2/20 0.46
NUAK1 O60285 3/20 0.40
FLT4 P35916 1/20 0.39
AURKA O14965 1/20 0.39
JAK3 P52333 6/20 0.39
JAK2 O60674 5/20 0.39
JAK1 P23458 4/20 0.39
TYK2 P29597 3/20 0.39
IKBKE Q14164 1/20 0.39
TBK1 Q9UHD2 1/20 0.39
AURKC Q9UQB9 1/20 0.38
IGF1R P08069 1/20 0.38
MAP4K1 Q92918 1/20 0.38
F11 P03951 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30956407 0.91 KDR (0.48) KDRAURKBNUAK1FLT4AURKA
SCHEMBL27059432 0.88 KDR (0.49) KDRAURKBFLT4AURKAJAK3
SCHEMBL28919841 0.86 JAK2 (0.40) NUAK1JAK3JAK2JAK1TYK2
SCHEMBL30956426 0.82 FLT4 (0.46) KDRAURKBNUAK1FLT4JAK3
SCHEMBL28606148 0.81 IGF1R (0.44) FLT4JAK3JAK2JAK1TYK2
SCHEMBL24852480 0.81 JAK3 (0.48) JAK3JAK2JAK1TYK2IGF1R
SCHEMBL30956612 0.80 JAK3 (0.49) NUAK1FLT4JAK3JAK2JAK1
SCHEMBL30956449 0.80 KDR (0.45) KDRAURKBFLT4JAK3JAK2
Hydrochloric Acid SCHEMBL30956501 0.80 NUAK1 (0.55) KDRAURKBNUAK1FLT4JAK3
SCHEMBL22098030 0.79 JAK2 (0.44) KDRFLT4JAK3JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118290403-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-07-05 CN disclosed
CN-113227074-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl derivatives, compositions and methods 凌科药业(杭州)有限公司 2021-08-06 CN disclosed