SCHEMBL28598985

SCHEMBL28598985

Fc1ccc(-c2cnc3[nH]ccc3c2Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.53
PRKCI P41743 2/20 0.53
RPS6KA3 P51812 4/20 0.51
MAPK1 P28482 1/20 0.48
MAPK14 Q16539 7/20 0.46
CSNK1D P48730 2/20 0.46
MAPK11 Q15759 1/20 0.46
CLK2 P49760 2/20 0.43
DYRK1A Q13627 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
DYRK1B Q9Y463 2/20 0.43
CLK1 P49759 1/20 0.43
DYRK2 Q92630 1/20 0.43
TRPA1 O75762 1/20 0.42
NUDT1 P36639 2/20 0.41
EGFR P00533 2/20 0.41
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30173343 1.00 AXL (0.53) AXLPRKCIRPS6KA3MAPK1MAPK14
SCHEMBL30173316 0.84 AXL (0.61) AXLPRKCIRPS6KA3CLK2DYRK1A
SCHEMBL28609163 0.84 AXL (0.61) AXLPRKCIRPS6KA3CLK2DYRK1A
SCHEMBL30173305 0.84 JAK2 (0.58) AXLPRKCIRPS6KA3MAPK1CLK2
SCHEMBL3725709 0.84 JAK2 (0.58) AXLPRKCIRPS6KA3MAPK1CLK2
SCHEMBL28596894 0.84 RPS6KA3 (0.49) AXLPRKCIRPS6KA3CLK2DYRK1A
SCHEMBL28596900 0.84 AXL (0.49) AXLPRKCIRPS6KA3CLK2DYRK1A
SCHEMBL30173331 0.84 AXL (0.49) AXLPRKCIRPS6KA3CLK2DYRK1A
SCHEMBL30173298 0.84 RPS6KA3 (0.49) AXLPRKCIRPS6KA3CLK2DYRK1A
SCHEMBL30173308 0.81 AXL (0.53) AXLPRKCIMAPK1DYRK1ACLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200983-B Compound with pyrrolopyridine structure, preparation method and medical application 中国药科大学 2023-01-03 CN disclosed
CN-113200983-A Compound with pyrrolopyridine structure, preparation method and medical application 中国药科大学 2021-08-03 CN disclosed