SCHEMBL28600429

SCHEMBL28600429

COc1cc(OC)cc(Oc2ccc(C(=O)O)cc2)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.70
CA2 P00918 1/20 0.70
RXRA P19793 2/20 0.68
KDM4E B2RXH2 1/20 0.59
PARP10 Q53GL7 2/20 0.58
PARP15 Q460N3 1/20 0.58
SRD5A2 P31213 3/20 0.56
ALDH1A1 P00352 2/20 0.54
RAB9A P51151 3/20 0.53
NPC1 O15118 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
POLB P06746 1/20 0.53
RXRB P28702 1/20 0.53
RXRG P48443 1/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
TTR P02766 1/20 0.51
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2511835 0.90 CA1 (0.87) CA1CA2RXRAKDM4EPARP10
SCHEMBL29531785 0.90 PARP10 (0.69) CA1CA2RXRAPARP10PARP15
SCHEMBL1877592 0.87 CA1 (0.63) CA1CA2RXRAKDM4ESRD5A2
SCHEMBL28060732 0.86 KMT2A (0.66) CA1CA2RXRAPARP10PARP15
SCHEMBL14811923 0.85 AKR1C3 (0.62) CA1CA2RXRASRD5A2ALDH1A1
SCHEMBL9702751 0.85 KDM4E (0.77) CA1CA2RXRAKDM4EPARP10
P-Anisic Acid SCHEMBL1157044 0.83 CA1 (1.00) CA1CA2RXRAKDM4EPARP10
P-Anisic Acid SCHEMBL43335 0.83 CA1 (1.00) CA1CA2RXRAKDM4EPARP10
Ethane SCHEMBL11219716 0.83 PARP10 (0.72) CA1CA2RXRAPARP10PARP15
Terephthalic Acid SCHEMBL9861713 0.83 PARP10 (0.78) CA1CA2RXRAPARP10PARP15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113045494-B Pyridone derivative and application thereof in preparation of drugs for preventing and/or treating tuberculosis caused by mycobacterium tuberculosis 四川大学华西医院 2022-04-26 CN disclosed
CN-113045494-A Pyridone derivative and application thereof in preparation of drugs for preventing and/or treating tuberculosis caused by mycobacterium tuberculosis 四川大学华西医院 2021-06-29 CN disclosed