SCHEMBL28600504

SCHEMBL28600504

[c]1coc(-n2ccnc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.38
LMNA P02545 3/20 0.36
MAPT P10636 2/20 0.36
ENPP2 Q13822 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
NOTUM Q6P988 1/20 0.36
CYP2A6 P11509 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
IDO1 P14902 2/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
CYP1A2 P05177 3/20 0.33
CYP2D6 P10635 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2C19 P33261 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
USP2 O75604 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23783439 0.68 CYP3A4 (0.41) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL28767572 0.67 CYP3A4 (0.39) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL28943672 0.67 CYP3A4 (0.39) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL6597600 0.65 CYP3A4 (0.39) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL15219432 0.64 CYP3A4 (0.37) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL16923117 0.64 CYP3A4 (0.54) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL1916742 0.61 CYP3A4 (0.38) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL20357191 0.61 LMNA (0.40) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL29131511 0.61 CYP3A4 (0.38) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL244552 0.61 CYP3A4 (0.38) CYP3A4LMNAMAPTENPP2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103582642-B HSP90 inhibitor 索隆-基特林癌症研究协会 2021-05-11 CN disclosed