SCHEMBL28601014

SCHEMBL28601014

O=CNOC(=O)[C@@H]1CN(c2cc(Cl)ncn2)CCO1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.35
EIF2AK4 Q9P2K8 1/20 0.35
KMO O15229 1/20 0.34
EGFR P00533 2/20 0.33
ERBB3 P21860 2/20 0.33
SCN9A Q15858 2/20 0.33
ELOVL1 Q9BW60 1/20 0.32
USP30 Q70CQ3 3/20 0.32
P4HTM Q9NXG6 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ATM Q13315 1/20 0.32
MAPK14 Q16539 1/20 0.32
FPR2 P25090 1/20 0.32
RAB9A P51151 1/20 0.31
MAP2K7 O14733 1/20 0.31
CYP2C19 P33261 1/20 0.30
LRRK2 Q5S007 1/20 0.30
PIK3CD O00329 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20899405 0.85 SCN9A (0.42) MAP4K4EIF2AK4KMOSCN9AELOVL1
SCHEMBL22873464 0.85 SCN9A (0.42) MAP4K4EIF2AK4KMOSCN9AELOVL1
SCHEMBL20899406 0.85 SCN9A (0.42) MAP4K4EIF2AK4KMOSCN9AELOVL1
SCHEMBL28607925 0.81 KMO (0.44) MAP4K4EIF2AK4KMOEGFRERBB3
SCHEMBL21797145 0.81 KMO (0.44) MAP4K4EIF2AK4KMOEGFRERBB3
Formamide SCHEMBL28601016 0.80 KMO (0.40) MAP4K4EIF2AK4KMOEGFRERBB3
SCHEMBL18399166 0.79 GRIN2B (0.43) MAP4K4USP30PIK3CD
SCHEMBL21796661 0.79 GRIN2B (0.43) MAP4K4USP30PIK3CD
SCHEMBL21796840 0.79 GRIN2B (0.43) MAP4K4USP30PIK3CD
SCHEMBL23525833 0.70 LRRK2 (0.47) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137510-B Compound (I) 葛兰素史密斯克莱知识产权发展有限公司 2021-07-20 CN disclosed