SCHEMBL28601809

SCHEMBL28601809

Cn1cc(C#Cc2n[nH]c3nc[nH]c(=O)c23)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 1/20 0.37
HAO1 Q9UJM8 2/20 0.36
GRM5 P41594 2/20 0.36
ACACB O00763 1/20 0.34
LCK P06239 1/20 0.34
RET P07949 1/20 0.34
SRC P12931 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
ADORA2A P29274 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRA1A P35348 1/20 0.33
XDH P47989 1/20 0.33
RAB9A P51151 1/20 0.33
BLM P54132 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LRRK2 Q5S007 1/20 0.31
DYRK1A Q13627 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28599648 0.77 IP6K1 (0.48) GRM5SRCLMNATSHRADORA2A
SCHEMBL28917753 0.77 DYRK1A (0.32) LMNATSHRADORA2ASLC6A4ADRA1A
SCHEMBL28918223 0.76 DYRK1A (0.38) ALDH1A1LMNATSHRADORA2ASLC6A4
SCHEMBL28918230 0.76 KDM4A (0.38) LMNATSHRADORA2ASLC6A4ADRA1A
SCHEMBL28608978 0.76 PIK3CA (0.39) HAO1GRM5LMNATSHRADORA2A
SCHEMBL28595680 0.74 PIK3CA (0.45) HAO1GRM5DYRK1A
SCHEMBL12540751 0.71 ACHE (0.35) ALDH1A1LMNATSHRADORA2ASLC6A4
SCHEMBL12541355 0.70 ACHE (0.34) ALDH1A1LMNATSHRADORA2ASLC6A4
SCHEMBL28590000 0.70 DYRK1A (0.35) ALDH1A1LMNATSHRADORA2ASLC6A4
SCHEMBL30947487 0.70 DYRK1A (0.40) ALDH1A1LMNATSHRADORA2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113880842-A Substituted alkynyl heterocyclic compounds 首药控股(北京)有限公司 2022-01-04 CN disclosed
CN-113004282-A Substituted alkynyl heterocyclic compounds 首药控股(北京)有限公司 2021-06-22 CN disclosed