SCHEMBL28603832

SCHEMBL28603832

COS(=O)(=O)Cc1cc(Br)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 2/20 0.34
SLC22A12 Q96S37 1/20 0.34
HTT P42858 1/20 0.33
NOS3 P29474 2/20 0.33
NOS1 P29475 2/20 0.33
NOS2 P35228 2/20 0.33
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
CDK2 P24941 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28358032 0.84 SMN1; SMN2 (0.34) SMN1; SMN2KDM4EALDH1A1TSHRSLC22A12
SCHEMBL28470585 0.81 KDM4E (0.41) SMN1; SMN2KDM4EALDH1A1HTTNOS3
SCHEMBL9988870 0.81 SLC22A12 (0.40) SMN1; SMN2KDM4EALDH1A1TSHRSLC22A12
SCHEMBL1662137 0.75 GBA1 (0.40) KDM4EALDH1A1TSHRMAPT
SCHEMBL31419110 0.75 GBA1 (0.40) KDM4EALDH1A1TSHRMAPT
SCHEMBL29049963 0.74 LMNA (0.46) ALDH1A1MEN1KMT2A
SCHEMBL12434098 0.73 KDM4E (0.37) SMN1; SMN2KDM4EALDH1A1NOS3NOS1
SCHEMBL28847152 0.72
SCHEMBL28381226 0.71 NPSR1 (0.33) ALDH1A1CDK2MAPT
SCHEMBL15526300 0.71 SLC22A12 (0.41) SMN1; SMN2KDM4EALDH1A1TSHRSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112812105-B Aminopyridyloxy pyrazole derivative, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2025-04-01 CN disclosed
CN-112812105-A Aminopyridyloxypyrazole derivative and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2021-05-18 CN disclosed