SCHEMBL28606145

SCHEMBL28606145

CC(C#N)NC(=O)c1ccccc1-c1nc(Nc2cnn(C3CCN(C)CC3)c2)ncc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 4/20 0.49
CDK4 P11802 2/20 0.49
CDK6 Q00534 2/20 0.49
CCNA2 P20248 1/20 0.49
FLT4 P35916 7/20 0.48
KDR P35968 5/20 0.48
JAK3 P52333 2/20 0.47
JAK2 O60674 1/20 0.47
JAK1 P23458 1/20 0.47
DDR2 Q16832 2/20 0.45
MAPK6 Q16659 1/20 0.44
CDK1 P06493 3/20 0.44
IGF1R P08069 3/20 0.44
CDK8 P49336 1/20 0.44
CDK7 P50613 1/20 0.44
CDK9 P50750 1/20 0.44
KCNH2 Q12809 1/20 0.44
MAP3K14 Q99558 1/20 0.43
PIK3CD O00329 1/20 0.42
CSF1R P07333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28612508 0.92 FLT4 (0.49) CDK2FLT4KDRJAK3JAK2
SCHEMBL28612506 0.91 FLT4 (0.55) CDK2FLT4KDRJAK3CDK1
SCHEMBL29942188 0.87 CDK4 (0.54) CDK2CDK4CDK6CCNA2FLT4
SCHEMBL28600652 0.87 CDK4 (0.54) CDK2CDK4CDK6CCNA2FLT4
SCHEMBL22097751 0.87 CDK4 (0.54) CDK2CDK4CDK6CCNA2FLT4
SCHEMBL29942180 0.87 CDK4 (0.54) CDK2CDK4CDK6CCNA2FLT4
SCHEMBL22089701 0.87 CDK4 (0.54) CDK2CDK4CDK6CCNA2FLT4
SCHEMBL30956508 0.85 JAK3 (0.54) CDK2CDK4CDK6CCNA2FLT4
SCHEMBL28598992 0.85 IGF1R (0.54) CDK2FLT4CDK1IGF1RCDK8
SCHEMBL28603799 0.84 IGF1R (0.46) CDK2FLT4KDRJAK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227074-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl derivatives, compositions and methods 凌科药业(杭州)有限公司 2021-08-06 CN disclosed