SCHEMBL28610085

SCHEMBL28610085

CC(C)(C)OC(=O)N[C@@H]1CCCN(c2ncc(Cl)cc2C(F)(F)F)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 3/20 0.54
JAK3 P52333 2/20 0.54
SYK P43405 2/20 0.48
MAP4K4 O95819 2/20 0.47
PDE10A Q9Y233 1/20 0.47
AURKA O14965 3/20 0.44
PDPK1 O15530 3/20 0.44
AURKB Q96GD4 3/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
EGFR P00533 1/20 0.42
LCK P06239 1/20 0.42
F10 P00742 1/20 0.42
RET P07949 1/20 0.42
ITGB2 P05107 1/20 0.41
ICAM1 P05362 1/20 0.41
ITGAL P20701 1/20 0.41
OPRK1 P41145 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31124490 1.00 BTK (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL28610086 1.00 BTK (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL28614144 0.85 JAK3 (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL28605629 0.85 JAK3 (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL28605626 0.85 JAK3 (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL31124509 0.85 JAK3 (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL31124452 0.85 JAK3 (0.54) BTKJAK3SYKMAP4K4PDE10A
SCHEMBL28610070 0.83 BTK (0.40) BTKJAK3MEN1KMT2AOPRK1
SCHEMBL28610069 0.83 BTK (0.40) BTKJAK3MEN1KMT2AOPRK1
SCHEMBL31124491 0.82 SYK (0.55) BTKJAK3SYKMAP4K4PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164461-A Heterocyclic derivatives as Nav1.7 and Nav1.8 blockers 拉夸里亚创药株式会社 2021-07-23 CN disclosed