SCHEMBL28611014

SCHEMBL28611014

O=C(O)CCCCCCNC(=O)N1CCC(N(c2ccccc2)c2cccc(F)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CHRM4 P08173 2/20 0.43
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
NPC1 O15118 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
CCR5 P51681 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18263850 0.92 HDAC6 (0.46) NAMPTMEN1KMT2ACYP2C9CYP2C19
SCHEMBL28601830 0.91 NAMPT (0.45) NAMPTMEN1KMT2ACYP2C19CHRM4
SCHEMBL18263775 0.91 MEN1 (0.44) NAMPTMEN1KMT2ACYP2C9CYP2C19
SCHEMBL28599106 0.86 NAMPT (0.50) NAMPTCHRM4DRD2DRD3ITGB3
SCHEMBL18271365 0.83 NAMPT (0.45) NAMPTDRD2DRD3CCR5
SCHEMBL18263694 0.82 HDAC6 (0.48) NAMPTHDAC6
SCHEMBL18263813 0.82 NAMPT (0.44) NAMPTMEN1KMT2ACYP2C19CHRM4
SCHEMBL18263786 0.81 HDAC6 (0.53) NAMPTHDAC6
SCHEMBL18263714 0.81 NAMPT (0.48) NAMPTDRD2DRD3OPRM1OPRD1
SCHEMBL28598203 0.78 CCR5 (0.49) MEN1KMT2ANPC1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026057-B Heterocycloalkyl-derived compounds as selective histone deacetylase inhibitors and pharmaceutical compositions containing the same 株式会社钟根堂 2021-08-06 CN disclosed