SCHEMBL28611990

SCHEMBL28611990

CC(C)(C)OC(=O)C1CCC2(CC1)CN(C(=O)OC(C)(C)C)c1ncccc12

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.46
CHRM4 P08173 3/20 0.41
CHRM1 P11229 2/20 0.41
KDM1A O60341 1/20 0.40
GPR119 Q8TDV5 3/20 0.38
POLB P06746 1/20 0.37
NOTUM Q6P988 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6002678 0.84 KCNH2 (0.43) KCNH2CHRM4CHRM1KDM1AGPR119
SCHEMBL7569116 0.79 KDM1A (0.47) KCNH2CHRM4CHRM1KDM1AGPR119
SCHEMBL23570520 0.79 POLB (0.43) KCNH2CHRM4KDM1AGPR119POLB
SCHEMBL20631821 0.73 POLB (0.38) KCNH2KDM1AGPR119POLB
SCHEMBL23570688 0.73 POLB (0.38) KCNH2CHRM4KDM1AGPR119POLB
SCHEMBL20631860 0.72 KDM1A (0.39) KCNH2CHRM4KDM1AGPR119POLB
SCHEMBL20632140 0.72 JAK1 (0.39) KDM1AGPR119POLB
SCHEMBL30968406 0.71 KDM1A (0.39) KCNH2CHRM4CHRM1KDM1AGPR119
SCHEMBL20630932 0.71 POLB (0.36) KCNH2CHRM4KDM1AGPR119POLB
SCHEMBL31505870 0.70 SLC18A3 (0.44) KCNH2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113015526-A Spirocyclic 2, 3-dihydro-7-azaindole compounds and uses thereof 豪夫迈·罗氏有限公司 2021-06-22 CN disclosed