SCHEMBL28612213

SCHEMBL28612213

Clc1cc(Cl)c2c(c1)C1(CCCCC1)CCO2

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.38
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
MAP3K14 Q99558 1/20 0.31
AKR1B1 P15121 1/20 0.31
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23668822 0.81 PDE7A (0.33) PDE7A
SCHEMBL28617434 0.77 PDE7A (0.38) PDE7ASLC6A4AHR
SCHEMBL6605186 0.70 AKR1B1 (0.42) PDE7AMAP3K14AKR1B1
SCHEMBL6605188 0.70 AKR1B1 (0.42) PDE7AMAP3K14AKR1B1
SCHEMBL6580397 0.70 AKR1B1 (0.42) PDE7AMAP3K14AKR1B1
SCHEMBL11345300 0.68 AKR1B1 (0.60) AKR1B1
SCHEMBL6760984 0.67 AKR1B1 (0.37) MAP3K14AKR1B1
SCHEMBL6605516 0.67 AKR1B1 (0.37) MAP3K14AKR1B1
SCHEMBL8793427 0.66 AKR1B1 (0.47) AKR1B1
SCHEMBL768845 0.64 MAP3K14 (0.32) MAP3K14AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113087700-B Spirocyclic tetrahydroquinazolines 苏州亚盛药业有限公司 2023-03-14 CN disclosed
CN-113087700-A Spirocyclic tetrahydroquinazolines 苏州亚盛药业有限公司 2021-07-09 CN disclosed