SCHEMBL28612475

SCHEMBL28612475

CC(C)(C)OC(=O)N[C@H]1CCc2sc(NC(=O)[C@H]3C[C@@H]3F)cc2C1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.36
BTK Q06187 1/20 0.36
KDM1A O60341 1/20 0.35
MAOB P27338 1/20 0.35
ABL1 P00519 3/20 0.35
CTSK P43235 2/20 0.34
DRD2 P14416 3/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
NAMPT P43490 1/20 0.32
JAK2 O60674 3/20 0.32
JAK1 P23458 3/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21603867 0.87 TP53 (0.39) EPHX2BTKKDM1AMAOBCTSK
SCHEMBL27415413 0.85 EPHX2 (0.36) EPHX2BTKKDM1AMAOBCTSK
SCHEMBL27415382 0.84 ABL1 (0.34) ABL1NPC1RAB9A
SCHEMBL31563954 0.78 EPHX2 (0.43) EPHX2BTKKDM1AMAOBCTSK
SCHEMBL31564173 0.77 EPHX2 (0.43) EPHX2BTKKDM1AMAOBCTSK
SCHEMBL28607624 0.76 ALDH1A1 (0.38) BTKKMT2ARAB9A
Trifluoroacetic Acid SCHEMBL28611854 0.74 ABL1 (0.36) ABL1
SCHEMBL28615820 0.72 MAPT (0.49) KMT2A
SCHEMBL28613536 0.72 MAPT (0.49) KMT2A
SCHEMBL29371263 0.72 NPC1 (0.47) EPHX2DRD2KMT2AL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112566910-A Thiophene derivatives for the treatment of IgE induced diseases UCB生物制药有限责任公司 2021-03-26 CN disclosed