SCHEMBL28614130

SCHEMBL28614130

COC(=O)c1cnc(N2CCCN(Cc3ccc(C(F)(F)F)cc3)CC2)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.49
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
HIF1A Q16665 2/20 0.46
EPAS1 Q99814 2/20 0.46
HRH3 Q9Y5N1 1/20 0.46
CHKA P35790 1/20 0.46
PPARD Q03181 1/20 0.46
PPARA Q07869 1/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28920588 0.91 SCD (0.52) SCDHDAC3HDAC4HDAC1HDAC7
SCHEMBL4804346 0.82 ALDH1A1 (0.61) SCDHDAC3HDAC4HDAC1HDAC7
SCHEMBL12933726 0.80 PARP1 (0.45) SCDHDAC3HDAC4HDAC1HDAC7
SCHEMBL1065675 0.80 GPR6 (0.50) SCDHRH3ALDH1A1PRKAA2PARP1
SCHEMBL31599315 0.79 HIF1A (0.41) HIF1AEPAS1PPARDPPARAKDM4E
SCHEMBL4087735 0.79 SCD (0.77) SCDKDM4EALDH1A1MEN1MAPT
SCHEMBL4812703 0.78 HDAC3 (0.78) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28619735 0.78 HDAC3 (0.49) SCDHDAC3HDAC4HDAC1HDAC7
SCHEMBL28619734 0.78 HDAC3 (0.49) SCDHDAC3HDAC4HDAC1HDAC7
SCHEMBL20176409 0.76 HRH3 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072546-A Five-membered heteroaromatic derivative and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed