SCHEMBL28614283

SCHEMBL28614283

Brc1cnc2[nH]cc(-c3ccncc3)c2c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.75
DYRK1A Q13627 2/20 0.75
PLK4 O00444 1/20 0.75
AURKA O14965 1/20 0.75
ROCK2 O75116 1/20 0.75
PRKD3 O94806 1/20 0.75
MAP4K4 O95819 1/20 0.75
PRKCG P05129 1/20 0.75
INSR P06213 1/20 0.75
CDK1 P06493 1/20 0.75
FES P07332 1/20 0.75
IGF1R P08069 1/20 0.75
ROS1 P08922 1/20 0.75
FGFR1 P11362 1/20 0.75
PHKG2 P15735 1/20 0.75
FER P16591 1/20 0.75
FLT1 P17948 1/20 0.75
CDK2 P24941 1/20 0.75
MARK3 P27448 1/20 0.75
FLT4 P35916 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1516750 0.86 JAK2 (1.00) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL28603325 0.85 DYRK1A (0.67) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL15333224 0.84 DYRK1A (0.74) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL1516629 0.83 DYRK1A (0.73) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL28595754 0.82 DYRK1A (0.63) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL28603327 0.82 DYRK1A (0.63) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL17952128 0.81 NTRK1 (0.62) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL17952449 0.81 NTRK1 (0.77) DYRK1ANTRK1PIK3CASLC2A1IMPDH2
SCHEMBL28610224 0.80 DYRK1A (0.68) JAK2DYRK1APLK4AURKAROCK2
SCHEMBL3765160 0.79 CDK8 (0.85) NTRK1PIK3CAAXLCDK8TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113214247-A Azaindole derivative marrow cell proliferation inhibitor, preparation method and application thereof in pharmacy 复旦大学 2021-08-06 CN disclosed