SCHEMBL28614964

SCHEMBL28614964

O=C(CCCCCCNC(=O)N1CCc2c([nH]c3ccccc23)C1)NO

nearest known ligand 0.78

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.78
HDAC1 Q13547 2/20 0.78
KMT2A Q03164 1/20 0.61
DRD2 P14416 2/20 0.58
DRD3 P35462 2/20 0.58
GPX4 P36969 1/20 0.57
TRPV1 Q8NER1 13/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28617480 0.92 KMT2A (0.73) HDAC6HDAC1KMT2ADRD2DRD3
SCHEMBL28920591 0.90 KMT2A (0.63) HDAC6HDAC1KMT2ADRD2DRD3
SCHEMBL8252701 0.88 HDAC6 (1.00) HDAC6HDAC1GPX4TRPV1
SCHEMBL997520 0.85 KMT2A (0.78) HDAC6HDAC1KMT2ADRD2DRD3
SCHEMBL998500 0.84 KMT2A (0.84) HDAC6HDAC1KMT2ADRD2DRD3
SCHEMBL28606538 0.82 KMT2A (0.76) HDAC6HDAC1KMT2ADRD2DRD3
SCHEMBL5787110 0.81 HDAC1 (0.74) HDAC6HDAC1
SCHEMBL998353 0.81 KMT2A (0.71) HDAC6HDAC1KMT2ADRD2DRD3
SCHEMBL1000934 0.80 GPX4 (0.63) KMT2AGPX4TRPV1
SCHEMBL999152 0.80 KMT2A (0.72) KMT2ADRD2DRD3GPX4TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121527-B Tricyclic compounds and uses thereof 上海辉启生物医药科技有限公司 2024-09-06 CN disclosed
CN-113121527-A Tricyclic compound and use thereof 上海辉启生物医药科技有限公司 2021-07-16 CN disclosed