SCHEMBL28618201

SCHEMBL28618201

N#Cc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(O)c(O)c(O)c3)C(C(=O)NCc3ccc4ccccc4c3)C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.44
F10 P00742 2/20 0.44
ADAM17 P78536 2/20 0.42
ALDH1A1 P00352 2/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 2/20 0.38
CA9 Q16790 2/20 0.38
MCHR1 Q99705 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
MC4R P32245 1/20 0.37
EIF2AK3 Q9NZJ5 1/20 0.37
GAA P10253 1/20 0.37
TGM2 P21980 1/20 0.37
CASR P41180 1/20 0.37
KAT6A Q92794 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28608791 0.88 HTT (0.47) ADAM17GAA
SCHEMBL26673483 0.85 F2 (0.45) F2F10ADAM17ALDH1A1KMT2A
SCHEMBL28618856 0.84 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1USP2GAA
SCHEMBL28618855 0.82 MAPT (0.46) ADAM17ALDH1A1CA1CA2CA4
SCHEMBL29720620 0.79 F10 (0.41) F2F10CA1CA2CA4
SCHEMBL26673511 0.79 F10 (0.45) F2F10ALDH1A1USP2GAA
SCHEMBL30608846 0.79 F10 (0.45) F2F10ALDH1A1USP2GAA
SCHEMBL26673510 0.79 F2 (0.48) F2F10ADAM17ALDH1A1CA1
SCHEMBL26673488 0.77 ALDH1A1 (0.53) F2F10ADAM17ALDH1A1KMT2A
SCHEMBL28601239 0.77 HTT (0.49) ALDH1A1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105395-B 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN disclosed