SCHEMBL28620033

SCHEMBL28620033

FC(F)(F)c1ccc(N2CCc3ccccc3C2)c(C#Cc2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
GAA P10253 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
BACE1 P56817 1/20 0.44
MAPK1 P28482 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 1/20 0.43
AKR1C3 P42330 1/20 0.38
NOTUM Q6P988 1/20 0.36
HSD17B3 P37058 1/20 0.36
GRM2 Q14416 1/20 0.36
GRM5 P41594 2/20 0.36
PKM P14618 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPN6 P29350 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28921827 0.83 BACE1 (0.46) MAPTKDM4EMEN1NPC1GAA
SCHEMBL3485666 0.77 ALDH1A1 (0.56) MAPTKDM4EMEN1NPC1GAA
SCHEMBL3484761 0.72 MAPT (0.64) MAPTMEN1RAB9AKMT2ANPSR1
SCHEMBL12204277 0.70 MAPT (0.47) MAPTKDM4EMEN1NPC1GAA
SCHEMBL30101923 0.70 EED (0.63) MAPTKDM4EMEN1NPC1GAA
SCHEMBL28626119 0.70 EED (0.63) MAPTKDM4EMEN1NPC1GAA
SCHEMBL10539432 0.70 ALDH1A1 (0.79) MAPTKDM4ENPSR1BACE1ALDH1A1
SCHEMBL14106286 0.69 ALDH1A1 (0.64) MAPTKDM4EMEN1NPC1GAA
SCHEMBL14106282 0.68 ALDH1A1 (0.75) MAPTKDM4EMEN1KMT2ANPSR1
SCHEMBL1922380 0.68 PTGDR2 (0.50) MEN1KMT2AALDH1A1GRM5PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307769-A 1-alkynyl tetrahydroisoquinoline compound and preparation method thereof 长江师范学院 2021-08-27 CN disclosed